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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T14987 | CMP8 | Estrogen Receptor/ERR , Estrogen/progestogen Receptor | |
CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM , 41 nM, 1100 nM and 2200 nM for MGERα, MGRERα, hERα and hERβ, res... |